SCHEMBL7380885

SCHEMBL7380885

NC(=O)C[CH]Cc1cc(Cl)cc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 3/20 0.38
HTR3B O95264 3/20 0.38
HTR3A P46098 3/20 0.38
HTR3D Q70Z44 3/20 0.38
HTR3C Q8WXA8 3/20 0.38
IDO1 P14902 5/20 0.36
EPHX1 P07099 1/20 0.36
TPMT P51580 1/20 0.34
KDM4E B2RXH2 2/20 0.34
SLC9A1 P19634 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
ADRA1D P25100 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33
ITGB3 P05106 1/20 0.32
ITGAV P06756 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417345 0.81 MEN1 (0.38) IDO1EPHX1
SCHEMBL7379832 0.77 PRSS1 (0.42) IDO1EPHX1TPMTSLC9A1ALDH1A1
SCHEMBL7377171 0.74 HTT (0.46) KDM4EALDH1A1GAA
SCHEMBL7386500 0.73 IDO1 (0.42) IDO1EPHX1GAA
SCHEMBL3340425 0.73 CA2 (0.46) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL27630839 0.72 IDO1 (0.45) IDO1EPHX1
Hydrochloric Acid SCHEMBL3341453 0.71 IDO1 (0.45) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL5215999 0.71 CA2 (0.55) HTR3AIDO1KDM4EALDH1A1
SCHEMBL4068734 0.69 CAPN1 (0.46) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL2654048 0.69 TSHR (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165500-A1 AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES,TNF-ALPHA,AND AGGRECANASE Du Pont Pharmaceuticals Company (US) 2002-01-02 EP disclosed
WO-2000059874-A1 NOVEL AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES, TNF-α, AND AGGRECANASE DU PONT PHARMACEUTICALS COMPANY (US) 2000-10-12 WO disclosed