SCHEMBL7382437

SCHEMBL7382437

CC(C)Oc1ccc(-c2ccc3ncc4cncn4c3n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
WDR5 P61964 1/20 0.37
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
MCL1 Q07820 2/20 0.35
ADORA2A P29274 1/20 0.35
DYRK1A Q13627 3/20 0.34
MAP4K4 O95819 1/20 0.34
DYRK2 Q92630 2/20 0.33
CLK1 P49759 1/20 0.33
BMPR1B O00238 1/20 0.32
ACVR1B P36896 1/20 0.32
ACVRL1 P37023 1/20 0.32
ACVR1 Q04771 1/20 0.32
ACP1 P24666 1/20 0.32
PIK3CD O00329 1/20 0.32
PIP5K1C O60331 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PI4KA P42356 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19781576 0.75 DYRK1A (0.50) WDR5TP53MAPTMCL1DYRK1A
SCHEMBL19781531 0.68 DYRK1A (0.45) MAPTDYRK1AATM
SCHEMBL21449908 0.68 DYRK1A (0.55) MAPTMCL1DYRK1APIM3ATM
SCHEMBL19781550 0.65 FDPS (0.40) CYP1A2WDR5TP53MAPTMCL1
SCHEMBL21449929 0.64 GABRP (0.45) DYRK1APIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL31140240 0.63 CYP2D6 (0.59) CYP1A2WDR5TP53MAPTMCL1
SCHEMBL14988627 0.62 MAP4K4 (0.46) CYP1A2WDR5TP53MAPTMCL1
SCHEMBL19781608 0.62 FGFR1 (0.46) CYP1A2MAPTDYRK1AATMMAOA
SCHEMBL25002926 0.61 MCL1 (0.43) CYP1A2WDR5TP53MAPTMCL1
SCHEMBL19781584 0.61 KDM4E (0.47) CYP1A2WDR5TP53MAPTMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993022314-A1 CERTAIN ARYL AND CYCLOALKYL FUSED IMIDAZOPYRAZINEDIONES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1993-11-11 WO disclosed