SCHEMBL7384200

SCHEMBL7384200

CCCCCOC(=O)c1cc2c(cn1)[nH]c1ccccc12

nearest known ligand 0.93

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.93
MAPT P10636 4/20 0.93
SMN1; SMN2 Q16637 3/20 0.93
KDM4E B2RXH2 3/20 0.93
CYP1A2 P05177 2/20 0.93
CYP3A4 P08684 2/20 0.93
HPGD P15428 2/20 0.93
CYP2C19 P33261 2/20 0.93
CYP2C9 P11712 1/20 0.93
TSHR P16473 1/20 0.93
GABRA1 P14867 12/20 0.84
GABRG2 P18507 12/20 0.84
GABRB3 P28472 12/20 0.84
GABRA5 P31644 12/20 0.84
GABRA3 P34903 12/20 0.84
GABRA2 P47869 12/20 0.84
GABRA6 Q16445 9/20 0.84
GABRA4 P48169 8/20 0.84
GABRP O00591 7/20 0.84
GABRD O14764 7/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2214572 0.96 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2
SCHEMBL29766941 0.96 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2
SCHEMBL2348263 0.92 GABRA1 (1.00) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2
SCHEMBL601711 0.87 GABRA1 (1.00) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2
SCHEMBL30274389 0.87 GABRA1 (1.00) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2
SCHEMBL29672619 0.87 GABRA1 (1.00) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2
SCHEMBL8146977 0.84 GABRA1 (0.78) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2
SCHEMBL7380516 0.84 GABRA1 (0.77) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2
Beta-Ccm SCHEMBL15648382 0.82 GABRA1 (0.91) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2
SCHEMBL31163651 0.82 GABRA1 (0.77) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5010077-A Tranquilizers A/S FERROSAN (DK) 1991-04-23 US disclosed
EP-0030254-B1 BETA-CARBOLIN-3-CARBOXYLIC ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR THERAPEUTICAL USE SCHERING AKTIENGESELLSCHAFT (DE) 1984-10-31 EP disclosed
US-4371536-A TRANQUILIZERS A/S FERROSAN (DK) 1983-02-01 US disclosed
EP-0030254-A1 Beta-carbolin-3-carboxylic acid derivatives, pharmaceutical compositions containing them and their therapeutical use SCHERING AKTIENGESELLSCHAFT (DE) 1981-06-17 EP disclosed