SCHEMBL7384253

SCHEMBL7384253

O=C(Cc1ccc(Cl)c(Cl)c1)N1CC2CC=CCC2C1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.59
SIGMAR1 Q99720 2/20 0.48
OPRK1 P41145 7/20 0.46
NPC1 O15118 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
NFKB1 P19838 1/20 0.46
CYP2C19 P33261 1/20 0.46
OPRD1 P41143 1/20 0.46
HIF1A Q16665 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
DRD4 P21917 1/20 0.45
SLC6A3 Q01959 1/20 0.45
TMEM97 Q5BJF2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7384247 1.00 KMT2A (0.59) KMT2ASIGMAR1OPRK1NPC1CYP1A2
SCHEMBL11687083 0.86 KMT2A (0.68) KMT2ASIGMAR1OPRK1NPC1CYP1A2
SCHEMBL16117817 0.81 OPRK1 (0.60) KMT2ASIGMAR1OPRK1NPC1CYP3A4
SCHEMBL5448229 0.79 KMT2A (0.58) KMT2ASIGMAR1OPRK1CYP3A4CYP2D6
SCHEMBL5448233 0.79 KMT2A (0.58) KMT2ASIGMAR1OPRK1CYP3A4CYP2D6
SCHEMBL24095117 0.75 KMT2A (0.73) KMT2ASIGMAR1OPRK1NPC1CYP1A2
SCHEMBL13504125 0.74 KMT2A (0.68) KMT2ASIGMAR1OPRK1NPC1CYP1A2
Hydrochloric Acid SCHEMBL7625422 0.72 KMT2A (0.69) KMT2ASIGMAR1OPRK1CYP1A2CYP2D6
SCHEMBL7379985 0.72 SIGMAR1 (0.63) SIGMAR1CYP1A2CYP2D6TMEM97
SCHEMBL7379983 0.72 SIGMAR1 (0.63) SIGMAR1CYP1A2CYP2D6TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409929-A Treating psychosis, dyskinesia THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-25 US disclosed
WO-1993016047-A1 HYDROISOINDOLINES AND HYDROISOQUINOLINES AS PSYCHOTROPIC DRUGS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-08-19 WO disclosed
US-5216018-A Antidyskinetic agents DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-06-01 US disclosed