SCHEMBL7385266

SCHEMBL7385266

CCOC(=O)NC(=N)c1ccc(CCc2nc3c(C)c(N(CC(=O)OC)S(=O)(=O)c4cccc5cccnc45)ccc3[nH]2)cc1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
F2 P00734 5/20 0.39
ALDH1A1 P00352 4/20 0.37
TSHR P16473 2/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 2/20 0.35
PKLR P30613 3/20 0.34
TP53 P04637 2/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7393934 0.89 F2 (0.49) F2ALDH1A1MAPTTP53POLB
SCHEMBL7395993 0.89 ALDH1A1 (0.37) F2ALDH1A1TSHRGAAMAPT
SCHEMBL7392529 0.82 TSHR (0.40) F2ALDH1A1TSHRGAAMAPT
SCHEMBL7395518 0.81 F2 (0.38) F2ALDH1A1TSHRGAAMAPT
SCHEMBL7391715 0.78 F2 (0.51) F2ALDH1A1MAPTTP53POLB
SCHEMBL6636191 0.78 F2 (0.68) F2ALDH1A1TSHRGAAMAPT
SCHEMBL7394301 0.77 F2 (0.50) F2ALDH1A1TSHRGAAMAPT
SCHEMBL7392579 0.77 F2 (0.45) F2ALDH1A1MAPTTP53POLB
SCHEMBL7392629 0.77 F2 (0.40) F2ALDH1A1TSHRGAAMAPT
SCHEMBL7388035 0.76 TSHR (0.38) F2ALDH1A1TSHRGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM ZENTRALE GMBH (DE) 2001-05-23 EP disclosed
WO-2000008014-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-02-17 WO disclosed