SCHEMBL7385447

SCHEMBL7385447

CCOC(=O)N1C2C=C(S(=O)(=O)C(F)(F)F)CC1CC2

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.42
CHRM1 P11229 9/20 0.36
TP53 P04637 2/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
GRM5 P41594 1/20 0.32
MAPT P10636 1/20 0.32
GPR119 Q8TDV5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3144755 0.81 CXCR3 (0.41) CXCR3CHRM1TP53CHRM4CHRM5
SCHEMBL13849989 0.74 CXCR3 (0.36) CXCR3TP53ALDH1A1TDP1
SCHEMBL29649963 0.72 DRD2 (0.35) CXCR3CHRM1
SCHEMBL11360845 0.71 CXCR3 (0.40) CXCR3CHRM1CHRM4CHRM5ALDH1A1
SCHEMBL14081576 0.70 SLC6A2 (0.46) CHRM1CHRM4CHRM5ALDH1A1TDP1
SCHEMBL20682190 0.69 CXCR3 (0.39) CXCR3CHRM1GPR119
SCHEMBL19014089 0.68 CXCR3 (0.38) CXCR3GPR119
SCHEMBL12094668 0.68 HTR2C (0.41)
SCHEMBL29336 0.68 CHRM2 (0.41) CHRM1GPR119
SCHEMBL41973 0.68 CHRM2 (0.41) CHRM1GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214303-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001016121-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF MERCK & CO., INC. (US) 2001-03-08 WO disclosed