SCHEMBL7387262

SCHEMBL7387262

Cc1nc(C#CC#C[Si](C)(C)C)cs1

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 18/20 0.51
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1243386 0.86 GRM5 (0.56) GRM5CYP1A2CYP2D6
SCHEMBL28749297 0.72
SCHEMBL18873238 0.69 GRM5 (0.54) GRM5CYP1A2CYP2D6
SCHEMBL1434084 0.69 GRM5 (0.63) GRM5CYP1A2CYP2D6
SCHEMBL29384255 0.69 GRM5 (0.63) GRM5CYP1A2CYP2D6
SCHEMBL4145767 0.69 GRM5 (0.72) GRM5CYP1A2CYP2D6
SCHEMBL15483095 0.68 GRM5 (0.53) GRM5CYP1A2CYP2D6
SCHEMBL22894216 0.68 GRM5 (0.51) GRM5CYP1A2CYP2D6
SCHEMBL3353813 0.68 GRM5 (0.68) GRM5CYP1A2CYP2D6
SCHEMBL6024302 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214303-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001016121-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF MERCK & CO., INC. (US) 2001-03-08 WO disclosed