SCHEMBL7387883

SCHEMBL7387883

CC(C)(C)[Si](C)(C)N1C(=O)CC1Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 2/20 0.39
ABCB1 P08183 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 2/20 0.39
USP2 O75604 1/20 0.39
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
GAA P10253 1/20 0.39
IDH1 O75874 2/20 0.36
RIPK1 Q13546 1/20 0.36
HPGD P15428 1/20 0.36
GRM2 Q14416 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7387880 1.00 TSHR (0.39) TSHRKMT2AALDH1A1ABCB1NPC1
SCHEMBL30259456 1.00 TSHR (0.39) TSHRKMT2AALDH1A1ABCB1NPC1
SCHEMBL10414651 0.79 GLA (0.43) TSHRKMT2AALDH1A1NPC1RAB9A
SCHEMBL6963830 0.76
SCHEMBL10660255 0.76
SCHEMBL6963835 0.76
SCHEMBL9815162 0.75 KMT2A (0.35) TSHRKMT2AALDH1A1NPC1RAB9A
SCHEMBL5156976 0.74 BRD4 (0.34)
SCHEMBL4098581 0.74 BRD4 (0.34)
SCHEMBL11003070 0.74 HCAR2 (0.42) ALDH1A1POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021405-B1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF HCMV INFECTIONS BOEHRINGER INGELHEIM CA LTD (CA) 2002-09-25 EP disclosed
US-6242439-B1 Azetidinone derivatives for the treatment of HCMV infections BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2001-06-05 US disclosed
EP-1021405-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF HCMV INFECTIONS BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2000-07-26 EP disclosed
WO-1999018072-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF HCMV INFECTIONS BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 1999-04-15 WO disclosed