SCHEMBL7388665

SCHEMBL7388665

NC1C(O)Cc2cc(C(=O)O)ccc2C1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
TDP1 Q9NUW8 3/20 0.41
KDM4E B2RXH2 6/20 0.40
MAPT P10636 3/20 0.40
POLB P06746 3/20 0.40
BLM P54132 1/20 0.40
GRM1 Q13255 1/20 0.40
MEN1 O00255 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM1A O60341 2/20 0.40
SRD5A2 P31213 4/20 0.37
SRD5A1 P18405 3/20 0.37
LTB4R Q15722 1/20 0.36
LTB4R2 Q9NPC1 1/20 0.36
PTPN1 P18031 1/20 0.35
GAA P10253 3/20 0.35
HSD17B10 Q99714 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7562014 0.76 TSHR (0.41) ALDH1A1KDM4EMAPTPOLBMEN1
SCHEMBL27796129 0.70 ALDH1A1 (0.46) ALDH1A1TDP1KDM4EMAPTPOLB
SCHEMBL13550403 0.69 ALDH1A1 (0.49) ALDH1A1TDP1KDM4EMAPTPOLB
SCHEMBL27775410 0.69 ALDH1A1 (0.44) ALDH1A1TDP1KDM4EMAPTPOLB
SCHEMBL8189658 0.69 ALDH1A1 (0.49) ALDH1A1TDP1KDM4EMAPTPOLB
SCHEMBL785696 0.69 ALDH1A1 (0.49) ALDH1A1TDP1KDM4EMAPTPOLB
Hydrochloric Acid SCHEMBL6642375 0.68 ALDH1A1 (0.52) ALDH1A1TDP1KDM4EMAPTPOLB
Hydrochloric Acid SCHEMBL785877 0.68 ALDH1A1 (0.47) ALDH1A1TDP1KDM4EMAPTPOLB
SCHEMBL29726906 0.67 ALDH1A1 (0.50) ALDH1A1TDP1KDM4EMAPTPOLB
SCHEMBL13163016 0.67 CHRNB2 (0.52) ALDH1A1TDP1KDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252178-A1 ALPHA-KETOAMIDE INHIBITORS OF HEPATITIS C VIRUS NS3 PROTEASE Bristol-Myers Squibb Pharma Company (US) 2002-10-30 EP disclosed
EP-1196436-A2 PEPTIDE BORONIC ACID INHIBITORS OF HEPATITIS C VIRUS PROTEASE Bristol-Myers Squibb Pharma Company (US) 2002-04-17 EP disclosed
WO-2001040262-A1 ALPHA-KETOAMIDE INHIBITORS OF HEPATITIS C VIRUS NS3 PROTEASE BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-06-07 WO disclosed
WO-2001002424-A2 PEPTIDE BORONIC ACID INHIBITORS OF HEPATITIS C VIRUS PROTEASE DU PONT PHARMACEUTICALS COMPANY (US) 2001-01-11 WO disclosed