SCHEMBL7389178

SCHEMBL7389178

COc1cc(N)c(Cl)cc1C(=O)NCC1CCN(CCCCCN(Cc2ccccc2)Cc2ccccc2)CC1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.69
DRD4 P21917 3/20 0.69
DRD3 P35462 3/20 0.69
HTR4 Q13639 15/20 0.65
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
ADRA2A P08913 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
ADRA2B P18089 1/20 0.56
ADRA2C P18825 1/20 0.56
ACHE P22303 1/20 0.56
SLC6A2 P23975 1/20 0.56
HTR2A P28223 1/20 0.56
HTR2C P28335 1/20 0.56
ADRA1A P35348 1/20 0.56
OPRK1 P41145 1/20 0.56
HTR2B P41595 1/20 0.56
CHRNA4 P43681 1/20 0.56
HTR3A P46098 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7380916 0.96 DRD2 (0.66) DRD2DRD4DRD3HTR4CYP1A2
SCHEMBL7385847 0.96 DRD2 (0.66) DRD2DRD4DRD3HTR4CYP1A2
SCHEMBL7385680 0.95 DRD2 (0.65) DRD2DRD4DRD3HTR4
SCHEMBL7393581 0.95 DRD2 (0.67) DRD2DRD4DRD3HTR4CYP1A2
SCHEMBL7390834 0.94 DRD2 (0.62) DRD2DRD4DRD3HTR4
SCHEMBL7390486 0.93 DRD2 (0.68) DRD2DRD4DRD3HTR4
SCHEMBL7393905 0.91 DRD2 (0.65) DRD2DRD4DRD3HTR4CYP1A2
SCHEMBL7391065 0.90 HTR4 (0.63) DRD2DRD4DRD3HTR4
SCHEMBL7392591 0.89 HTR4 (0.62) DRD2DRD4DRD3HTR4
SCHEMBL7389865 0.89 HTR4 (0.63) DRD2DRD4DRD3HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5864039-A THERAPEUTIC TREATMENT OF VARIOUS GASTROINTESTINAL DISEASES, CENTRAL NERVOUS DISORDERS, CARDIOVASCULAR DISORDERS, URINARY DISEASES, UROGENITAL DISORDERS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1999-01-26 US disclosed
EP-0873990-A1 BENZOIC ACID COMPOUNDS AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1998-10-28 EP disclosed