SCHEMBL7390002

SCHEMBL7390002

COc1cccc(-c2nc3ccccc3[nH]2)c1OC(=O)C(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 2/20 0.58
RAB9A P51151 3/20 0.50
NPC1 O15118 2/20 0.50
KMT2A Q03164 2/20 0.47
HPSE Q9Y251 1/20 0.47
PARP1 P09874 2/20 0.47
KDM4E B2RXH2 2/20 0.47
PDE5A O76074 2/20 0.46
PARP2 Q9UGN5 1/20 0.46
SLC2A1 P11166 1/20 0.46
GUSB P08236 1/20 0.46
HDAC6 Q9UBN7 1/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
USP2 O75604 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7396331 0.86 KDM4E (0.53) AMY1ARAB9ANPC1KDM4EPDE5A
SCHEMBL7395552 0.83 PARP1 (0.59) AMY1ARAB9ANPC1KMT2AHPSE
SCHEMBL7992209 0.80 AMY1A (0.43) AMY1ARAB9ANPC1KMT2AKDM4E
SCHEMBL7394125 0.77 AMY1A (0.54) AMY1ARAB9ANPC1KMT2AHPSE
SCHEMBL2096956 0.77 AMY1A (0.76) AMY1ARAB9ANPC1PARP1KDM4E
SCHEMBL31027930 0.77 AMY1A (0.76) AMY1ARAB9ANPC1PARP1KDM4E
SCHEMBL31429666 0.76 AMY1A (0.71) AMY1ARAB9ANPC1KMT2AKDM4E
SCHEMBL7393458 0.76 AMY1A (0.71) AMY1ARAB9ANPC1KMT2AKDM4E
SCHEMBL7398763 0.76 AMY1A (0.50) AMY1ARAB9ANPC1KDM4EALDH1A1
SCHEMBL7389695 0.75 PARP1 (0.51) AMY1ARAB9ANPC1KMT2AHPSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001066526-A1 ESTER DERIVATIVES OF DIMETHYLPROPIONIC ACID AND PHARMACETUICAL COMPOSITIONS CONTAINING THEM CERMOL S.A. (CH) 2001-09-13 WO claimed
EP-1132381-A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them CERMOL S.A. (CH) 2001-09-12 EP claimed
EP-1132381-A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them CERMOL S.A. (CH) 2001-09-12 EP disclosed