SCHEMBL739128

SCHEMBL739128

CC(C)c1ccc2nc([C@@H]3CCCN(C(=O)C[C@@H](Cc4ccc5ccccc5c4)N(C(=O)O)C(C)(C)C)C3)[nH]c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.46
GRIN2B Q13224 1/20 0.45
CYP1A2 P05177 3/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2C19 P33261 3/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PPARA Q07869 1/20 0.40
KDM4E B2RXH2 8/20 0.40
POLB P06746 4/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
LMNA P02545 2/20 0.38
USP2 O75604 1/20 0.38
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
ALDH1A1 P00352 1/20 0.37
BCL9 O00512 1/20 0.36
CTNNB1 P35222 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741506 0.90 MAPK1 (0.44) MAPK1GRIN2BCYP1A2CYP3A4CYP2C19
SCHEMBL741405 0.85 CYP1A2 (0.42) MAPK1GRIN2BCYP1A2CYP3A4CYP2C19
SCHEMBL741843 0.85 PTGS1 (0.51) MAPK1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL741796 0.83 HPGD (0.42) MAPK1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL740770 0.83 HTR2B (0.49) MAPK1GRIN2BCYP1A2CYP3A4CYP2C19
SCHEMBL740304 0.82 GRIN2B (0.50) MAPK1GRIN2BCYP1A2CYP3A4CYP2C19
SCHEMBL739281 0.82 POLB (0.46) MAPK1GRIN2BCYP1A2CYP3A4CYP2C19
SCHEMBL740023 0.82 GRIN2B (0.50) MAPK1GRIN2BCYP1A2CYP3A4CYP2C19
SCHEMBL741088 0.82 HTR2B (0.39) MAPK1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL762864 0.82 MAPK1 (0.45) MAPK1GRIN2BCYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed