SCHEMBL741405

SCHEMBL741405

CC(C)(C)N(C(=O)O)[C@@H](CC(=O)N1CCC[C@@H](c2nc3cc([N+](=O)[O-])ccc3[nH]2)C1)Cc1ccc2ccccc2c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAPK1 P28482 1/20 0.40
TACR1 P25103 5/20 0.39
KDM4E B2RXH2 5/20 0.38
POLB P06746 3/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
GRIN2B Q13224 1/20 0.38
CASR P41180 2/20 0.38
CTNNB1 P35222 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741506 0.94 MAPK1 (0.44) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL739128 0.85 MAPK1 (0.46) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL741843 0.83 PTGS1 (0.51) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL763211 0.82 CYP1A2 (0.41) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL741796 0.81 HPGD (0.42) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL740770 0.81 HTR2B (0.49) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL744560 0.81 HRH1 (0.37) CYP2D6SMN1; SMN2TACR1KMT2ACASR
SCHEMBL740023 0.81 GRIN2B (0.50) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL740304 0.81 GRIN2B (0.50) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL739281 0.81 POLB (0.46) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed