SCHEMBL7394254

SCHEMBL7394254

COc1cc(C(NC(C)=O)C2CCN(C(CC(=O)O)c3ccccc3)C2)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 12/20 0.47
ITGA4 P13612 12/20 0.47
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
CCR5 P51681 1/20 0.38
CCR3 P51677 1/20 0.38
GAA P10253 1/20 0.38
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7432396 0.95 ITGB1 (0.48) ITGB1ITGA4MEN1KMT2ACCR3
SCHEMBL7392592 0.92 ITGB1 (0.50) ITGB1ITGA4MEN1KMT2AGAA
SCHEMBL7393051 0.91 ITGB1 (0.47) ITGB1ITGA4MEN1KMT2AGAA
SCHEMBL7429588 0.89 ITGB1 (0.51) ITGB1ITGA4MEN1KMT2AGAA
SCHEMBL7535883 0.86 ITGA4 (0.46) ITGB1ITGA4MEN1KMT2ACCR3
SCHEMBL7426846 0.85 ITGB1 (0.51) ITGB1ITGA4MEN1KMT2AGAA
SCHEMBL7394287 0.85 ITGA4 (0.50) ITGB1ITGA4MEN1KMT2AALDH1A1
SCHEMBL7425026 0.84 ITGB1 (0.47) ITGB1ITGA4MEN1KMT2ACCR3
SCHEMBL7425213 0.84 ITGB1 (0.49) ITGB1ITGA4MEN1KMT2AGAA
SCHEMBL7388792 0.84 ITGB1 (0.46) ITGB1ITGA4MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999054321-A1 SUBSTITUTED DIAMINES AND THEIR USE AS CELL ADHESION INHIBITORS AVENTIS PHARMA LIMITED (GB) 1999-10-28 WO disclosed