SCHEMBL7429588

SCHEMBL7429588

COc1cc(C(NC(C)=O)C2CCN(C(C)CC(=O)O)CC2)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 15/20 0.51
ITGA4 P13612 15/20 0.51
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
LPAR1 Q92633 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7392592 0.95 ITGB1 (0.50) ITGB1ITGA4MEN1KMT2AALDH1A1
SCHEMBL7428230 0.93 ITGB1 (0.53) ITGB1ITGA4MEN1KMT2AALDH1A1
SCHEMBL7432396 0.92 ITGB1 (0.48) ITGB1ITGA4MEN1KMT2AALDH1A1
SCHEMBL7393051 0.90 ITGB1 (0.47) ITGB1ITGA4MEN1KMT2AGAA
SCHEMBL7383245 0.90 ITGB1 (0.49) ITGB1ITGA4MEN1KMT2AALDH1A1
SCHEMBL7394254 0.89 ITGB1 (0.47) ITGB1ITGA4MEN1KMT2AALDH1A1
SCHEMBL7425047 0.88 ITGB1 (0.54) ITGB1ITGA4MEN1KMT2AMAPT
SCHEMBL7428883 0.87 ITGB1 (0.50) ITGB1ITGA4MEN1KMT2AALDH1A1
SCHEMBL7392261 0.87 THRB (0.47) ITGB1ITGA4MEN1KMT2AALDH1A1
SCHEMBL7394287 0.86 ITGA4 (0.50) ITGB1ITGA4MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999054321-A1 SUBSTITUTED DIAMINES AND THEIR USE AS CELL ADHESION INHIBITORS AVENTIS PHARMA LIMITED (GB) 1999-10-28 WO disclosed