SCHEMBL739451

SCHEMBL739451

CC(=O)NCCn1c([C@@H]2CCCN(C(=O)C[C@H](N)Cc3ccc(-c4cnc(N)nc4)cc3)C2)nc2c(C)cccc21

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 2/20 0.34
DPP4 P27487 3/20 0.33
CYP2D6 P10635 2/20 0.32
HRH1 P35367 2/20 0.32
ALOX5AP P20292 1/20 0.32
BTK Q06187 2/20 0.31
NPY1R P25929 2/20 0.31
NMT1 P30419 1/20 0.31
CFD P00746 1/20 0.31
PROKR1 Q8TCW9 2/20 0.30
KCNH2 Q12809 1/20 0.30
HPGDS O60760 1/20 0.30
KDM4E B2RXH2 1/20 0.30
TP53 P04637 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739453 1.00 MAP3K12 (0.34) MAP3K12DPP4CYP2D6HRH1ALOX5AP
SCHEMBL742198 0.95 CPB1 (0.33) MAP3K12DPP4CYP2D6HRH1ALOX5AP
SCHEMBL742197 0.95 CPB1 (0.33) MAP3K12DPP4CYP2D6HRH1ALOX5AP
SCHEMBL740085 0.93 DPP4 (0.33) DPP4CYP2D6HRH1BTKNPY1R
SCHEMBL739670 0.93 DPP4 (0.33) DPP4CYP2D6HRH1BTKNPY1R
SCHEMBL741102 0.93 NMT1 (0.34) MAP3K12DPP4CYP2D6HRH1ALOX5AP
SCHEMBL738711 0.93 NMT1 (0.34) MAP3K12DPP4CYP2D6HRH1ALOX5AP
SCHEMBL739266 0.90 HRH1 (0.42) CYP2D6HRH1PROKR1KCNH2
SCHEMBL739267 0.90 HRH1 (0.42) CYP2D6HRH1PROKR1KCNH2
SCHEMBL743557 0.87 CD274 (0.35) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed