SCHEMBL7395299

SCHEMBL7395299

Nc1c(Cl)cc(C(=O)O)c2c1C=CCO2

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.33
POLB P06746 3/20 0.33
TSHR P16473 2/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 3/20 0.32
GAA P10253 1/20 0.32
HTR4 Q13639 2/20 0.31
ALDH1A1 P00352 3/20 0.31
TP53 P04637 1/20 0.31
CASP1 P29466 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
HTR3A P46098 1/20 0.31
HTR3D Q70Z44 1/20 0.31
HTR3C Q8WXA8 1/20 0.31
KDM4E B2RXH2 2/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5759463 0.74 TSHR (0.37) POLBTSHRMAPTALDH1A1TP53
SCHEMBL7333144 0.74 KDM4E (0.37) POLBCYP3A4MAPTGAAALDH1A1
SCHEMBL505507 0.73 HTR4 (0.41) HTTPOLBTSHRCYP3A4MAPT
SCHEMBL2944408 0.73 HTR4 (0.50) HTTPOLBTSHRCYP3A4HTR4
SCHEMBL1502018 0.70 HTR4 (0.51) HTR4HTR3EHTR3BHTR3AHTR3D
SCHEMBL6823514 0.69 CA1 (0.34) CA1CA2CA9
SCHEMBL5316552 0.68 HTR4 (0.47) HTR4HTR3EHTR3BHTR3AHTR3D
SCHEMBL7333211 0.67 HTR4 (0.46) HTR4HTR3EHTR3BHTR3AHTR3D
SCHEMBL8948599 0.66 CA1 (0.31) CA1CA2CA9
SCHEMBL7411412 0.65 HTT (0.34) HTTPOLBTSHRCYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5502209-A SIDE EFFECT REDUCTION, GASTROINTESTINAL SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1996-03-26 US disclosed
EP-0691341-A1 Benzopyrancarboxamide derivatives, salt thereof, process for the preparation of same and use thereof SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1996-01-10 EP disclosed