SCHEMBL7396138

SCHEMBL7396138

O=C(O)/C=C/c1ccc2ccccc2c1Br

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.65
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
TBXA2R P21731 1/20 0.48
PTGER4 P35408 1/20 0.48
PTGFR P43088 1/20 0.48
PTGER3 P43115 1/20 0.48
PTGER2 P43116 1/20 0.48
PTGDR Q13258 1/20 0.48
HDAC8 Q9BY41 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
NFKB1 P19838 1/20 0.47
CA4 P22748 1/20 0.47
POLB P06746 1/20 0.46
EIF2AK2 P19525 1/20 0.45
CSNK2A2 P19784 1/20 0.45
CSNK2B P67870 1/20 0.45
CSNK2A1 P68400 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7396139 1.00 MAOB (0.65) MAOBKDM4ELMNATBXA2RPTGER4
SCHEMBL7394709 0.81 MAOB (0.59) MAOBKDM4EHDAC8HDAC6POLB
SCHEMBL7394712 0.81 MAOB (0.59) MAOBKDM4EHDAC8HDAC6POLB
SCHEMBL8746644 0.81 KDM4E (0.50) MAOBKDM4ELMNATBXA2RPTGER4
SCHEMBL765995 0.81 CYP1B1 (0.54) MAOBKDM4ELMNATBXA2RPTGER4
SCHEMBL765996 0.81 CYP1B1 (0.54) MAOBKDM4ELMNATBXA2RPTGER4
SCHEMBL21662321 0.80 MAOB (0.78) MAOBKDM4ELMNAHDAC8HDAC6
SCHEMBL28723354 0.79 MAOB (0.67) MAOBNFKB1CYP1A1CYP1B1RAB9A
SCHEMBL600540 0.79 HDAC8 (0.67) KDM4EHDAC8HDAC6CA1CA2
SCHEMBL29404405 0.79 HDAC8 (0.67) KDM4EHDAC8HDAC6CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288261-B1 DRUGS FOR INHIBITION OF ENZYMES ABBOTT LABORATORIES 2001-09-11 US disclosed
WO-2000037433-A1 INHIBITORS OF MATRIX METALLOPROTEINASES ABBOTT LABORATORIES (US) 2000-06-29 WO disclosed