SCHEMBL7396195

SCHEMBL7396195

O=C(O)c1ccccc1C(=O)Nc1nc2c([nH]1)c(=O)n(CC1CC1)c(=O)n2CC1CC1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 0.52
PDE4B Q07343 8/20 0.52
PDE4C Q08493 8/20 0.52
PDE4D Q08499 8/20 0.52
PDE5A O76074 7/20 0.52
ADORA1 P30542 6/20 0.45
ADORA2A P29274 3/20 0.45
ADORA2B P29275 3/20 0.45
ADORA3 P0DMS8 1/20 0.45
PCK1 P35558 4/20 0.45
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7393964 0.89 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7502502 0.84 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7436271 0.72 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7026234 0.68 PDE4A (0.70) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7809025 0.68 PDE4A (0.70) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7395897 0.67 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9427714 0.64 ADORA2A (0.69) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7398584 0.64 PDE4A (0.64) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL8102407 0.64 ADORA2B (0.43) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL11705400 0.63 NPC1 (0.74) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550559-A1 XANTHINES Beecham Group p.l.c. (GB) 1993-07-14 EP claimed
WO-1992005176-A1 XANTHINES BEECHAM GROUP PLC (GB) 1992-04-02 WO claimed
WO-1992005176-A1 XANTHINES BEECHAM GROUP PLC (GB) 1992-04-02 WO disclosed