SCHEMBL7436271

SCHEMBL7436271

CC(C)(C)Nc1nc2c([nH]1)c(=O)n(CC1CC1)c(=O)n2CC1CC1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 9/20 0.69
PDE4B Q07343 9/20 0.69
PDE4C Q08493 9/20 0.69
PDE4D Q08499 9/20 0.69
PDE5A O76074 8/20 0.69
ADORA1 P30542 8/20 0.51
ADORA2A P29274 4/20 0.47
ADORA2B P29275 4/20 0.47
SIRT1 Q96EB6 1/20 0.47
SIRT3 Q9NTG7 1/20 0.47
SIRT5 Q9NXA8 1/20 0.47
ADORA3 P0DMS8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13986122 0.86 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL13986185 0.83 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9502308 0.77 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7026234 0.76 PDE4A (0.70) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7809025 0.76 PDE4A (0.70) PDE4APDE4BPDE4CPDE4DPDE5A
Cipamfylline SCHEMBL26990 0.76 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7395750 0.75 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL13986119 0.75 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7395897 0.74 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7025747 0.74 ADORA1 (0.64) PDE4APDE4BPDE4CPDE4DPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550559-A1 XANTHINES Beecham Group p.l.c. (GB) 1993-07-14 EP claimed
WO-1992005176-A1 XANTHINES BEECHAM GROUP PLC (GB) 1992-04-02 WO claimed
EP-0550559-A1 XANTHINES Beecham Group p.l.c. (GB) 1993-07-14 EP disclosed
WO-1992005176-A1 XANTHINES BEECHAM GROUP PLC (GB) 1992-04-02 WO disclosed