SCHEMBL739762

SCHEMBL739762

COCCCn1c(C2CCCN(C(=O)CC(Cc3ccc(-c4ccc(C(=O)OC)cc4Cl)cc3)NC(=O)OC(C)(C)C)C2)nc2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 4/20 0.38
AGTR1 P30556 3/20 0.38
HRH1 P35367 8/20 0.37
CYP2D6 P10635 6/20 0.37
KCNH2 Q12809 7/20 0.36
PROKR1 Q8TCW9 1/20 0.35
CHRM1 P11229 3/20 0.35
DRD2 P14416 1/20 0.35
TBXA2R P21731 1/20 0.35
TP53 P04637 1/20 0.35
MMP3 P08254 1/20 0.34
MMP7 P09237 1/20 0.34
MMP10 P09238 1/20 0.34
MMP12 P39900 1/20 0.34
PADI4 Q9UM07 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739761 1.00 AGTR2 (0.38) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL741086 0.95 AGTR2 (0.38) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL741085 0.95 AGTR2 (0.38) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL10292320 0.94 AGTR2 (0.37) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL763882 0.93 AGTR2 (0.37) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL763793 0.92 HRH1 (0.40) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL739120 0.92 HRH1 (0.39) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL739119 0.92 HRH1 (0.39) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL762929 0.89 KCNH2 (0.41) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL739547 0.89 HRH1 (0.41) HRH1CYP2D6KCNH2CHRM1PADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed