SCHEMBL763882

SCHEMBL763882

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc(-c4ccc(C(=O)NCCO)cc4Cl)cc3)NC(=O)OC(C)(C)C)C2)nc2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 4/20 0.37
AGTR1 P30556 3/20 0.37
HRH1 P35367 7/20 0.36
CYP2D6 P10635 6/20 0.36
KCNH2 Q12809 6/20 0.35
PTGER4 P35408 1/20 0.34
PROKR1 Q8TCW9 1/20 0.34
PPARG P37231 1/20 0.34
CHRM1 P11229 2/20 0.34
CNR2 P34972 1/20 0.33
MMP3 P08254 1/20 0.33
MMP7 P09237 1/20 0.33
MMP10 P09238 1/20 0.33
MMP12 P39900 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10292320 0.97 AGTR2 (0.37) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL739762 0.93 AGTR2 (0.38) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL741086 0.93 AGTR2 (0.38) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL739761 0.93 AGTR2 (0.38) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL741085 0.93 AGTR2 (0.38) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL763793 0.90 HRH1 (0.40) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL763247 0.90 KCNH2 (0.39) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL762735 0.90 HRH1 (0.38) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL741536 0.89 HRH1 (0.38) AGTR2AGTR1HRH1CYP2D6KCNH2
SCHEMBL741535 0.89 HRH1 (0.38) AGTR2AGTR1HRH1CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed