SCHEMBL7397697

SCHEMBL7397697

O=C1c2ccccc2C(=O)N1c1ccc2cccnc2c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.63
PSMD14 O00487 1/20 0.63
POLB P06746 1/20 0.63
MMP2 P08253 1/20 0.63
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
HTT P42858 2/20 0.49
ALDH1A1 P00352 5/20 0.45
KDM4E B2RXH2 3/20 0.45
GAA P10253 1/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 2/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
NR4A2 P43354 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CHRNA7 P36544 1/20 0.44
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19343024 0.78 ALDH1A1 (0.47) TP53PSMD14POLBMMP2MEN1
SCHEMBL18121475 0.77 POLB (0.84) TP53PSMD14POLBMMP2MEN1
SCHEMBL3179738 0.72 TSHR (0.57) POLBKMT2AHTTALDH1A1KDM4E
SCHEMBL3186382 0.72 TSHR (0.57) POLBKMT2AHTTALDH1A1KDM4E
SCHEMBL15836590 0.71 TP53 (0.55) TP53PSMD14POLBMMP2MEN1
SCHEMBL4649471 0.71 KMT2A (0.78) MEN1KMT2AHTTALDH1A1GAA
SCHEMBL5200701 0.70 KDM4E (0.54) TP53PSMD14POLBMMP2MEN1
SCHEMBL11705831 0.70 ALDH1A1 (0.50) TP53PSMD14POLBMMP2MEN1
SCHEMBL15000605 0.70 KMT2A (0.54) TP53POLBMEN1KMT2AALDH1A1
SCHEMBL3787691 0.70 CHRNA7 (0.48) TP53PSMD14POLBMMP2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM ZENTRALE GMBH (DE) 2001-05-23 EP disclosed
WO-2000008014-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-02-17 WO disclosed