SCHEMBL7398692

SCHEMBL7398692

O=C1C=Nc2ccccc2CC1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.48
NOS1 P29475 1/20 0.48
NOS2 P35228 1/20 0.48
TRPA1 O75762 11/20 0.47
CYP2A6 P11509 1/20 0.43
CES1 P23141 1/20 0.40
NPC1 O15118 3/20 0.38
RAB9A P51151 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.37
SRD5A1 P18405 1/20 0.36
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
MAPK14 Q16539 1/20 0.35
CYP1A2 P05177 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30804579 0.81 TRPA1 (0.59) NOS3NOS1NOS2TRPA1CYP2A6
SCHEMBL1119424 0.81 TRPA1 (0.59) NOS3NOS1NOS2TRPA1CYP2A6
SCHEMBL30804590 0.79 TRPA1 (0.57) NOS3NOS1NOS2TRPA1CYP2A6
Hydrochloric Acid SCHEMBL8588830 0.79 TRPA1 (0.57) TRPA1CYP2A6NPC1RAB9ACYP1A2
Hydrochloric Acid SCHEMBL8588251 0.79 TRPA1 (0.57) TRPA1CYP2A6NPC1RAB9ACYP1A2
SCHEMBL31145655 0.77 TRPA1 (0.70) NOS3NOS1NOS2TRPA1NPC1
Formic Acid SCHEMBL28613405 0.73 TRPA1 (0.50) TRPA1CYP2A6CYP1A2
SCHEMBL29910169 0.71 TRPA1 (0.47) TRPA1
SCHEMBL56649 0.70 NOS3 (0.52) NOS3NOS1NOS2TRPA1CYP2A6
SCHEMBL688175 0.69 NOS3 (0.56) NOS3NOS1NOS2TRPA1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0593603-B1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-11-20 EP disclosed
US-6127359-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 2000-10-03 US disclosed
US-5939412-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 1999-08-17 US disclosed
US-5693636-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 1997-12-02 US disclosed
EP-0593603-A1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1994-04-27 EP disclosed
WO-1993000095-A2 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1993-01-07 WO disclosed