SCHEMBL7399080

SCHEMBL7399080

O=C(C[C@H](F)C(=O)O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.69

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMO O15229 4/20 0.69
TSHR P16473 1/20 0.52
SLC6A4 P31645 1/20 0.49
SLC6A3 Q01959 1/20 0.49
HSD11B1 P28845 1/20 0.48
SRD5A2 P31213 1/20 0.46
POLB P06746 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
GRN P28799 1/20 0.44
SORT1 Q99523 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399077 1.00 KMO (0.69) KMOTSHRSLC6A4SLC6A3HSD11B1
SCHEMBL728316 1.00 KMO (0.69) KMOTSHRSLC6A4SLC6A3HSD11B1
SCHEMBL19642672 0.84 KMO (0.75) KMOTSHRSLC6A4SLC6A3HSD11B1
SCHEMBL3670103 0.81 KMO (0.71) KMOTSHRSLC6A4SLC6A3HSD11B1
SCHEMBL3670105 0.81 KMO (0.71) KMOTSHRSLC6A4SLC6A3HSD11B1
SCHEMBL4386002 0.81 KMO (1.00) KMOTSHRSLC6A4SLC6A3
SCHEMBL3676715 0.81 KMO (0.71) KMOTSHRSLC6A4SLC6A3HSD11B1
SCHEMBL728113 0.81 KMO (1.00) KMOTSHRSLC6A4SLC6A3
SCHEMBL3670421 0.81 KMO (1.00) KMOTSHRSLC6A4SLC6A3
SCHEMBL7797590 0.80 KMO (1.00) KMOTSHRSLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6323240-B1 HALOGENATED DERIVATIVES AS ENZYME INHIBITORS PHARMACIA & UPJOHN S.P.A. (IT) 2001-11-27 US disclosed
EP-0858443-A1 4-PHENYL-4-OXO-BUTANOIC ACID DERIVATIVES WITH KYNURENINE-3-HYDROXYLASE INHIBITING ACTIVITY PHARMACIA & UPJOHN S.p.A. (IT) 1998-08-19 EP disclosed
WO-1997017317-A1 4-PHENYL-4-OXO-BUTANOIC ACID DERIVATIVES WITH KYNURENINE-3-HYDROXYLASE INHIBITING ACTIVITY PHARMACIA & UPJOHN S.P.A. (IT) 1997-05-15 WO disclosed