SCHEMBL7399749

SCHEMBL7399749

CCO/C=C/C(=O)c1cccnc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 8/20 0.54
CYP1A2 P05177 8/20 0.54
CYP1B1 Q16678 8/20 0.54
CYP3A4 P08684 5/20 0.54
CYP2D6 P10635 5/20 0.54
MAPK1 P28482 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
GPR52 Q9Y2T5 1/20 0.51
MAPT P10636 3/20 0.50
KMT2A Q03164 3/20 0.50
CAPN1 P07384 1/20 0.50
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
MEN1 O00255 1/20 0.50
LMNA P02545 2/20 0.49
ALDH1A1 P00352 2/20 0.49
HPGD P15428 1/20 0.49
APP P05067 1/20 0.48
GSK3B P49841 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399751 1.00 CYP1A1 (0.54) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL27948287 0.81 HTT (0.53) CYP1A1CYP1A2CYP1B1CYP2D6NPSR1
SCHEMBL10275628 0.80 AKT1 (0.54) CYP1A2CYP1B1CYP3A4MAPK1NPSR1
SCHEMBL10275631 0.80 AKT1 (0.54) CYP1A2CYP1B1CYP3A4MAPK1NPSR1
SCHEMBL10439177 0.80 AKT1 (0.54) CYP1A2CYP1B1CYP3A4MAPK1NPSR1
SCHEMBL10036804 0.77 CYP1A1 (0.63) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL166048 0.77 CYP1A1 (0.63) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL7368740 0.76 MAPK1 (0.60) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL14305648 0.76 MAPT (0.57) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL7368742 0.76 MAPK1 (0.60) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed