SCHEMBL7399867

SCHEMBL7399867

CN1CCc2ccc(NC(=O)Nc3ccnc4ccccc34)cc2C1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.74
HTR2B P41595 8/20 0.74
ADRA2A P08913 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50
PLK4 O00444 1/20 0.47
CHEK1 O14757 1/20 0.47
PDPK1 O15530 1/20 0.47
PRKD3 O94806 1/20 0.47
MAP4K4 O95819 1/20 0.47
CHEK2 O96017 1/20 0.47
CDK1 P06493 1/20 0.47
PIM1 P11309 1/20 0.47
RPS6KB1 P23443 1/20 0.47
CDK2 P24941 1/20 0.47
FLT4 P35916 1/20 0.47
KDR P35968 1/20 0.47
CSNK1D P48730 1/20 0.47
CDK8 P49336 1/20 0.47
CLK2 P49760 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7663182 0.99 HTR2C (0.73) HTR2CHTR2BADRA2AADRA2BADRA2C
SCHEMBL7664641 0.85 HTR2B (1.00) HTR2CHTR2BADRA2AADRA2BADRA2C
SCHEMBL7664636 0.85 HTR2B (1.00) HTR2CHTR2BADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL7656658 0.84 HTR2B (0.98) HTR2CHTR2BADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL7656654 0.84 HTR2B (0.98) HTR2CHTR2BADRA2AADRA2BADRA2C
SCHEMBL8137589 0.83 KDM4E (0.56) HTR2CHTR2BNPC1RAB9A
SCHEMBL7654434 0.81 HTR2B (0.78) HTR2CHTR2BPLK4CHEK1PDPK1
Hydrochloric Acid SCHEMBL7658689 0.81 HTR2B (0.87) HTR2CHTR2BADRA2AADRA2BADRA2C
SCHEMBL8109950 0.80 HTR2C (0.67) HTR2CHTR2BADRA2AADRA2BADRA2C
SCHEMBL8130701 0.79 NPC1 (0.65) NPC1RAB9AABCB1ROCK2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003737-A1 PHENYL UREA AND PHENYL THIOUREA DERIVATIVES AS HFGAN72 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2000-05-31 EP disclosed
WO-1999009024-A1 PHENYL UREA AND PHENYL THIOUREA DERIVATIVES AS HFGAN72 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1999-02-25 WO disclosed