SCHEMBL7399887

SCHEMBL7399887

COc1cc(OC2CCN(C(=O)CC(C)(C)NC(=O)OC(C)(C)C)CC2)ccc1C(=O)N1CC[CH]CC1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OXTR P30559 10/20 0.43
AVPR2 P30518 2/20 0.43
AVPR1A P37288 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HSD11B1 P28845 1/20 0.41
HIF1A Q16665 1/20 0.39
PDE4B Q07343 3/20 0.39
PDE4A P27815 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
KMT2A Q03164 1/20 0.38
ERBB2 P04626 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7405740 0.84 OXTR (0.45) OXTRAVPR2AVPR1AALDH1A1HSD11B1
SCHEMBL7484095 0.81 OXTR (0.72) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL7508507 0.81 PDE4B (0.51) OXTRAVPR2AVPR1AALDH1A1HSD11B1
SCHEMBL7399308 0.79 OXTR (0.51) OXTRAVPR2AVPR1AALDH1A1HSD11B1
SCHEMBL7494734 0.77 OXTR (0.49) OXTRAVPR2AVPR1AALDH1A1HSD11B1
SCHEMBL7398524 0.76 OXTR (0.60) OXTRAVPR2AVPR1AALDH1A1HSD11B1
SCHEMBL7358039 0.73 GPR119 (0.53) ALDH1A1PDE4BPDE4APDE4CPDE4D
SCHEMBL30606457 0.73 GPR119 (0.53) ALDH1A1PDE4BPDE4APDE4CPDE4D
SCHEMBL18310133 0.72 GPR119 (0.54) ALDH1A1PDE4BPDE4APDE4CPDE4D
SCHEMBL7355186 0.72 GPR119 (0.54) ALDH1A1PDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714299-A4 1996-07-10 EP disclosed
EP-0714299-A1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO. INC. (US) 1996-06-05 EP disclosed
WO-1995002405-A1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1995-01-26 WO disclosed