SCHEMBL7399995

SCHEMBL7399995

CCCCS(=O)(=O)NC(CN(C=O)c1cc(OCCCNC2=NCCN2)no1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.43
ITGAV P06756 15/20 0.43
ITGB5 P18084 1/20 0.43
ITGB6 P18564 1/20 0.43
ITGA2B P08514 8/20 0.39
CHRM2 P08172 1/20 0.36
SLC6A4 P31645 1/20 0.36
WDR5 P61964 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399991 0.85 ITGB3 (0.38) ITGB3ITGAVITGA2BCHRM2SLC6A4
SCHEMBL7401924 0.85 ITGB3 (0.44) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL7399998 0.83 ITGB3 (0.51) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL8549170 0.82 ITGB3 (0.36) ITGB3ITGAVITGA2BCHRM2SLC6A4
Iodide SCHEMBL7403599 0.79 ITGB3 (0.49) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL7405166 0.77 ITGB3 (0.48) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL7354614 0.73 ITGB3 (0.46) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL7347851 0.73 ITGB3 (0.47) ITGB3ITGAVITGA2B
SCHEMBL7401916 0.71 ITGB3 (0.37) ITGB3ITGA2B
SCHEMBL7401929 0.70 ITGB3 (0.47) ITGB3ITGAVITGB5ITGB6ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO claimed
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO disclosed