SCHEMBL7401929

SCHEMBL7401929

CCCCOC(=O)NC(CNC(=O)c1cc(OCCCNC2=NCCN2)no1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.47
ITGAV P06756 17/20 0.47
ITGB5 P18084 1/20 0.44
ITGB6 P18564 1/20 0.44
SMPD1 P17405 1/20 0.40
ITGA2B P08514 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5027067 0.89 ITGB3 (0.60) ITGB3ITGAVITGB5ITGB6ITGA2B
Iodide SCHEMBL7403601 0.89 ITGB3 (0.60) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL6111422 0.89 ITGB3 (0.60) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL7401332 0.86 ITGB3 (0.59) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL7401335 0.86 ITGB3 (0.59) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL7399998 0.85 ITGB3 (0.51) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL13059980 0.84 ITGB3 (0.54) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL7982063 0.83 ITGB3 (0.42) ITGB3SMPD1ITGA2B
SCHEMBL7401924 0.83 ITGB3 (0.44) ITGB3ITGAVITGB5ITGB6ITGA2B
SCHEMBL7038265 0.80 ITGB3 (0.49) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP claimed
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO claimed
US-6214834-B1 ANGIOGENESIS INHIBITORS; ANTIINFLAMMATORY AGENTS; ANTICANCER AGENTS DUPONT PHARMACEUTICALS COMPANY 2001-04-10 US disclosed
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP disclosed
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO disclosed