SCHEMBL7400100

SCHEMBL7400100

COc1cc(OC2CCN(Cc3cc(C)nc(Cl)c3)CC2)ccc1C(=O)N1CC[CH]CC1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OXTR P30559 10/20 0.51
KMT2A Q03164 5/20 0.49
MEN1 O00255 4/20 0.49
ADRB2 P07550 3/20 0.44
AVPR2 P30518 1/20 0.43
AVPR1A P37288 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399308 0.78 OXTR (0.51) OXTRAVPR2AVPR1A
SCHEMBL7398524 0.75 OXTR (0.60) OXTRAVPR2AVPR1A
SCHEMBL7362816 0.75 OXTR (0.85) OXTRAVPR2AVPR1A
SCHEMBL7494734 0.74 OXTR (0.49) OXTRAVPR2AVPR1A
SCHEMBL7405740 0.73 OXTR (0.45) OXTRKMT2AAVPR2AVPR1A
SCHEMBL7508507 0.71 PDE4B (0.51) OXTRKMT2AMEN1AVPR2AVPR1A
SCHEMBL3882603 0.71 TSHR (0.60) OXTRKMT2AMEN1
SCHEMBL7399887 0.71 OXTR (0.43) OXTRKMT2AAVPR2AVPR1A
SCHEMBL7506857 0.69 MAPT (0.51) OXTRKMT2AMEN1AVPR2AVPR1A
SCHEMBL4750836 0.68 GAA (0.74) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714299-A4 1996-07-10 EP disclosed
EP-0714299-A1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO. INC. (US) 1996-06-05 EP disclosed
WO-1995002405-A1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1995-01-26 WO disclosed