SCHEMBL7400351

SCHEMBL7400351

CCCCN1CCC(Cn2c(C)cc(=O)n3c4ccccc4c(C(=O)O)c23)CC1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 1/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PMP22 Q01453 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GSK3B P49841 1/20 0.40
HRH2 P25021 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9342316 0.73 HTR4 (0.48) HTR4KDM4EALDH1A1PMP22NPSR1
SCHEMBL7400348 0.73 HTR4 (0.45) HTR4
SCHEMBL9341470 0.72 HTR4 (0.50) HTR4KDM4EALDH1A1PMP22NPSR1
SCHEMBL7331887 0.70 HRH2 (0.54) HRH2
Hydrochloric Acid SCHEMBL7422511 0.68 KDM4E (0.44) HTR4KDM4EALDH1A1PMP22NPSR1
SCHEMBL7360838 0.67 HTR4 (0.49) HTR4KDM4EALDH1A1PMP22NPSR1
SCHEMBL7383392 0.67 KCNH2 (0.51) KDM4E
Hydrochloric Acid SCHEMBL7537446 0.66 HTR4 (0.48) HTR4
SCHEMBL24380823 0.66 HTR4 (0.44) HTR4KDM4EALDH1A1
SCHEMBL9341292 0.66 KDM4E (0.49) KDM4EALDH1A1PMP22NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0662959-A1 5-HT4 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-07-19 EP claimed
WO-1994007859-A1 5-HT4 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-04-14 WO claimed
EP-0662959-A1 5-HT4 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-07-19 EP disclosed
WO-1994007859-A1 5-HT4 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-04-14 WO disclosed