SCHEMBL7360838

SCHEMBL7360838

CCCCN1CCC(CC2Cn3c(c(C(=O)O)c4ccccc43)S2)CC1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 4/20 0.49
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PMP22 Q01453 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9341470 0.74 HTR4 (0.50) HTR4KDM4EALDH1A1PMP22NPSR1
SCHEMBL9342316 0.73 HTR4 (0.48) HTR4KDM4EALDH1A1PMP22NPSR1
SCHEMBL7383392 0.69 KCNH2 (0.51) KDM4E
SCHEMBL8566824 0.69 HTR4 (0.47) HTR4KDM4EALDH1A1PMP22NPSR1
SCHEMBL7360842 0.69 KCNH2 (0.41) HTR4KDM4EALDH1A1PMP22NPSR1
SCHEMBL7331887 0.68 HRH2 (0.54)
SCHEMBL8574546 0.68 HTR4 (0.46) HTR4KDM4EALDH1A1PMP22NPSR1
SCHEMBL9341292 0.68 KDM4E (0.49) KDM4EALDH1A1PMP22NPSR1
SCHEMBL7421133 0.67 CHRM1 (0.42) HTR4
SCHEMBL7400351 0.67 HTR4 (0.43) HTR4KDM4EALDH1A1PMP22NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630376-A1 CONDENSED INDOLE DERIVATIVES AS 5HT 4?-RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-12-28 EP disclosed
WO-1993018036-A1 CONDENSED INDOLE DERIVATIVES AS 5HT4-RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-09-16 WO disclosed