SCHEMBL7401074

SCHEMBL7401074

Cc1cc(C)c(S(=O)(=O)NC(CNC(=O)C2CC(CCCC(=O)Nc3nc4ccccc4[nH]3)ON2)C(=O)O)c(C)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.52
ITGAV P06756 13/20 0.52
ITGA2B P08514 12/20 0.52
ITGB1 P05556 5/20 0.49
ITGA5 P08648 4/20 0.49
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7405983 0.90 ITGB3 (0.52) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7405357 0.88 ITGAV (0.49) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7401670 0.85 ITGB3 (0.70) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7401078 0.84 ITGB3 (0.74) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7406637 0.80 ITGB3 (0.52) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7982239 0.80 ITGAV (0.53) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7403054 0.80 ITGB3 (0.47) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7405451 0.79 ITGB3 (0.52) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7969330 0.79 ITGB3 (0.52) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL7400646 0.78 ITGB3 (0.53) ITGB3ITGAVITGA2BITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP claimed
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO claimed
US-6214834-B1 ANGIOGENESIS INHIBITORS; ANTIINFLAMMATORY AGENTS; ANTICANCER AGENTS DUPONT PHARMACEUTICALS COMPANY 2001-04-10 US disclosed
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP disclosed
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO disclosed