SCHEMBL7401778

SCHEMBL7401778

Cc1cc(C)c(S(=O)(=O)NC(CNC(=O)C2CC(CCCc3c[nH]c(N)n3)NO2)C(=O)O)c(C)c1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 16/20 0.51
ITGB3 P05106 15/20 0.51
ITGA2B P08514 15/20 0.51
ITGB1 P05556 2/20 0.39
ITGA5 P08648 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7402546 0.88 ITGAV (0.53) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7985868 0.85 ITGAV (0.47) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7985993 0.83 ITGB3 (0.52) ITGAVITGB3ITGA2B
SCHEMBL7407086 0.81 ITGB3 (0.46) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7402542 0.80 ITGB3 (0.77) ITGAVITGB3ITGA2B
SCHEMBL7402690 0.80 ITGAV (0.67) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7980567 0.80 ITGB3 (0.51) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7979032 0.80 ITGAV (0.51) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7986014 0.80 ITGB3 (0.67) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7402705 0.80 ITGB3 (0.48) ITGAVITGB3ITGA2BITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO claimed
US-6214834-B1 ANGIOGENESIS INHIBITORS; ANTIINFLAMMATORY AGENTS; ANTICANCER AGENTS DUPONT PHARMACEUTICALS COMPANY 2001-04-10 US disclosed
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP disclosed
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO disclosed