SCHEMBL740216

SCHEMBL740216

CC(C)(C)OC(=O)NC(CC(=O)O)Cc1ccncc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.55
CYP3A4 P08684 5/20 0.48
CYP17A1 P05093 1/20 0.47
APP P05067 4/20 0.46
CTSS P25774 5/20 0.44
CTSK P43235 4/20 0.44
CTSL P07711 1/20 0.44
CTSB P07858 1/20 0.44
ACE P12821 1/20 0.43
KLK5 Q9Y337 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740215 1.00 ATM (0.55) ATMCYP3A4CYP17A1APPCTSS
SCHEMBL1519945 0.88 ATM (0.70) ATMCYP3A4APPCTSSCTSK
SCHEMBL489490 0.88 ATM (0.70) ATMCYP3A4APPCTSSCTSK
SCHEMBL489489 0.88 ATM (0.70) ATMCYP3A4APPCTSSCTSK
SCHEMBL7639933 0.87 ATM (0.50) ATMCYP3A4CYP17A1APPCTSS
SCHEMBL4897776 0.86 ATM (0.54) ATMCYP3A4CYP17A1APPCTSS
SCHEMBL4899353 0.86 ATM (0.54) ATMCYP3A4CYP17A1APPCTSS
SCHEMBL7897952 0.85 ATM (0.56) ATMCYP3A4APPCTSSCTSK
SCHEMBL29163523 0.85 ATM (0.56) ATMAPPCTSSCTSKCTSL
SCHEMBL28132845 0.85 ATM (0.60) ATMAPPCTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed