SCHEMBL4899353

SCHEMBL4899353

CC(C)(C)OC(=O)N[C@@H](CO)Cc1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.54
CYP17A1 P05093 1/20 0.49
ROCK2 O75116 5/20 0.48
ROCK1 Q13464 5/20 0.48
PRKACA P17612 3/20 0.48
PRKX P51817 3/20 0.48
PRKG1 Q13976 3/20 0.48
CLK4 Q9HAZ1 3/20 0.48
MAPK1 P28482 3/20 0.48
IRAK1 P51617 2/20 0.48
PKN2 Q16513 2/20 0.48
RPS6KA5 O75582 2/20 0.48
RPS6KA4 O75676 2/20 0.48
GSK3B P49841 2/20 0.48
GSK3A P49840 1/20 0.48
SGK2 Q9HBY8 1/20 0.48
CYP3A4 P08684 6/20 0.47
LIMK1 P53667 2/20 0.46
RPS6KB1 P23443 1/20 0.46
PRKG2 Q13237 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4897776 1.00 ATM (0.54) ATMCYP17A1ROCK2ROCK1PRKACA
SCHEMBL740216 0.86 ATM (0.55) ATMCYP17A1CYP3A4APPCTSS
SCHEMBL740215 0.86 ATM (0.55) ATMCYP17A1CYP3A4APPCTSS
SCHEMBL271855 0.86 ATM (0.71) ATMMAPK1CYP3A4APPCTSS
SCHEMBL257912 0.86 ATM (0.71) ATMMAPK1CYP3A4APPCTSS
SCHEMBL1529562 0.86 ATM (0.71) ATMMAPK1CYP3A4APPCTSS
SCHEMBL6479279 0.84 CTSS (0.57) ATMMAPK1CYP3A4APPCTSS
SCHEMBL6479222 0.84 CTSS (0.57) ATMMAPK1CYP3A4APPCTSS
SCHEMBL21676555 0.84 ATM (0.55) ATMMAPK1CYP3A4APPCTSS
SCHEMBL6479218 0.84 CTSS (0.57) ATMMAPK1CYP3A4APPCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080242694-A1 Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith D SIDOCKY NEIL R 2008-10-02 US disclosed
CN-1202096-C 2-aminothiazoline derivatives and their use as no-synthase inhibitors AVENTIS PHARMA SA (FR) 2005-05-18 CN disclosed
CN-1444572-A 2-aminothiazoline derivatives and their use as no-synthase inhibitors AVENTIS PHARMA SA (FR) 2003-09-24 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242694-A1 Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith JAK2, CHEK2, MTOR ATM 45/4885CYP17A1 1806/4885ROCK2 1237/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.