SCHEMBL7402255

SCHEMBL7402255

O=C1CC(C(F)(F)F)=NN1Cc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.60
GAA P10253 1/20 0.60
THRB P10828 1/20 0.60
KDM4E B2RXH2 3/20 0.46
LMNA P02545 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
MAPT P10636 3/20 0.41
HPGD P15428 2/20 0.41
GSK3A P49840 2/20 0.41
GSK3B P49841 2/20 0.41
EHMT2 Q96KQ7 1/20 0.40
POLB P06746 2/20 0.40
HTT P42858 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
PDE3B Q13370 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL964206 0.76 ALDH1A1 (1.00) ALDH1A1GAATHRBKDM4ELMNA
SCHEMBL15057965 0.74 ALDH1A1 (0.64) ALDH1A1GAATHRBKDM4ELMNA
SCHEMBL1461002 0.73 GAA (0.37) ALDH1A1GAATHRBKDM4ETDP1
SCHEMBL178857 0.72 LOX (0.71) ALDH1A1GAAKDM4ETDP1MEN1
SCHEMBL3529328 0.72 ALDH1A1 (0.60) ALDH1A1GAATHRBKDM4ELMNA
SCHEMBL1754745 0.67 PGR (0.75) ALDH1A1GAATHRBKDM4ELMNA
SCHEMBL10080903 0.66 GAA (0.64) ALDH1A1GAATHRBKDM4ELMNA
SCHEMBL359249 0.66 ALDH1A1 (0.56) ALDH1A1GAATHRBKDM4ELMNA
SCHEMBL359250 0.66 ALDH1A1 (0.56) ALDH1A1GAATHRBKDM4ELMNA
SCHEMBL1758434 0.66 KDM4E (0.72) ALDH1A1GAATHRBKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750550-A RESPIRATORY SYSTEM DISORDERS SANOFI (FR) 1998-05-12 US disclosed
WO-1997010243-A1 2-(PYRAZOL-5-YL-OXYMETHYL)-1,2-BENZISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SANOFI (US) 1997-03-20 WO disclosed