SCHEMBL7403266

SCHEMBL7403266

Cc1cc(-c2nnc3c4ccccc4c(Cl)nn23)no1.Cc1cc(C(=O)O)no1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 5/20 0.50
GABRG2 P18507 5/20 0.50
GABRB3 P28472 5/20 0.50
GABRA5 P31644 5/20 0.50
GABRA3 P34903 5/20 0.50
GABRA2 P47869 5/20 0.50
GABRA4 P48169 1/20 0.50
GABRA6 Q16445 1/20 0.50
L3MBTL1 Q9Y468 2/20 0.47
RXFP1 Q9HBX9 1/20 0.47
CACNA2D1 P54289 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
RAB9A P51151 2/20 0.41
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
TP53 P04637 1/20 0.41
GFER P55789 1/20 0.41
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31058084 0.90 GABRA1 (0.58) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1258627 0.90 GABRA1 (0.58) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL2192508 0.83 RXFP1 (0.52) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7475422 0.78 GABRA1 (0.58) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL17364040 0.77 RXFP1 (0.49) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7478081 0.77 RXFP1 (0.52) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL12416449 0.76 RXFP1 (0.51) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7209133 0.76 GABRA1 (0.53) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7208520 0.76 GABRA1 (0.56) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7487597 0.75 GABRA1 (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002042305-A1 NITROGEN SUBSTITUTED 1,2,4-TRIAZOLO[3,4-A]PHTHALAZINE DERIVATIVES FOR ENHANCING COGNITION MERCK SHARP & DOHME LIMITED (GB) 2002-05-30 WO disclosed