SCHEMBL7404184

SCHEMBL7404184

Cc1cc(COc2ccc(N(CC(C)(O)C(=O)NO)C(=O)C(F)(F)F)cc2)c2ccccc2n1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 17/20 0.57
MMP2 P08253 3/20 0.47
MMP13 P45452 3/20 0.47
MMP9 P14780 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6597422 1.00 ADAM17 (0.57) ADAM17MMP2MMP13MMP9
SCHEMBL6597457 1.00 ADAM17 (0.57) ADAM17MMP2MMP13MMP9
SCHEMBL6597686 0.83 ADAM17 (0.53) ADAM17MMP2MMP13MMP9
SCHEMBL7450520 0.83 ADAM17 (0.53) ADAM17MMP2MMP13MMP9
SCHEMBL6600735 0.83 ADAM17 (0.53) ADAM17MMP2MMP13MMP9
Trifluoroacetic Acid SCHEMBL6597459 0.79 ADAM17 (0.57) ADAM17MMP2
Trifluoroacetic Acid SCHEMBL6597417 0.79 ADAM17 (0.57) ADAM17MMP2
SCHEMBL6596414 0.78 ADAM17 (0.62) ADAM17MMP2
SCHEMBL6593905 0.78 ADAM17 (0.62) ADAM17MMP2
SCHEMBL7402737 0.78 ADAM17 (0.62) ADAM17MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263756-A2 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA Bristol-Myers Squibb Pharma Company (US) 2002-12-11 EP disclosed
WO-2001070734-A2 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-09-27 WO disclosed