SCHEMBL740434

SCHEMBL740434

COCCCn1c(C2CC(C)CN(C(=O)C[C@H](N)Cc3ccc4ccccc4c3)C2)nc2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.38
HRH1 P35367 4/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 8/20 0.37
CHRM1 P11229 1/20 0.37
POLB P06746 2/20 0.37
USP2 O75604 1/20 0.37
TP53 P04637 6/20 0.37
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
THRB P10828 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740435 1.00 KCNH2 (0.38) KCNH2HRH1CYP2D6MAPTCHRM1
SCHEMBL762990 0.92 KCNH2 (0.39) KCNH2HRH1CYP2D6MAPTCHRM1
SCHEMBL739245 0.90 HRH1 (0.46) KCNH2HRH1CYP2D6CHRM1POLB
SCHEMBL739244 0.90 HRH1 (0.46) KCNH2HRH1CYP2D6CHRM1POLB
SCHEMBL763789 0.86 CTSB (0.37) KCNH2HRH1CYP2D6MAPTCHRM1
SCHEMBL741060 0.86 HRH1 (0.38) KCNH2HRH1CYP2D6MAPTCHRM1
SCHEMBL738317 0.83 HRH1 (0.39) KCNH2HRH1CYP2D6CHRM1
SCHEMBL740603 0.83 KCNH2 (0.43) KCNH2HRH1CYP2D6MAPTCHRM1
SCHEMBL740604 0.83 KCNH2 (0.43) KCNH2HRH1CYP2D6MAPTCHRM1
SCHEMBL740554 0.83 KCNH2 (0.39) KCNH2HRH1CYP2D6CHRM1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed