SCHEMBL7404607

SCHEMBL7404607

CNC(=O)c1cccc(NC(=O)Nc2ccnc3ccccc23)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 4/20 0.61
DNMT3A Q9Y6K1 4/20 0.61
CLK1 P49759 1/20 0.61
HTR2C P28335 8/20 0.58
HTR2B P41595 8/20 0.58
DNMT3L Q9UJW3 3/20 0.53
EHMT1 Q9H9B1 2/20 0.53
TRPV1 Q8NER1 1/20 0.52
GSK3A P49840 2/20 0.51
GSK3B P49841 2/20 0.51
PLK4 O00444 1/20 0.51
CHEK1 O14757 1/20 0.51
PDPK1 O15530 1/20 0.51
PRKD3 O94806 1/20 0.51
MAP4K4 O95819 1/20 0.51
CHEK2 O96017 1/20 0.51
CDK1 P06493 1/20 0.51
PIM1 P11309 1/20 0.51
RPS6KB1 P23443 1/20 0.51
CDK2 P24941 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7660465 0.99 DNMT1 (0.60) DNMT1DNMT3ACLK1HTR2CHTR2B
Hydrochloric Acid SCHEMBL7661070 0.88 CLK1 (0.61) DNMT1DNMT3ACLK1HTR2CHTR2B
Dimethylamine SCHEMBL7660199 0.82 HTR2C (0.72) DNMT1DNMT3AHTR2CHTR2BDNMT3L
Hydrochloric Acid SCHEMBL7652839 0.81 MAPT (0.60) HTR2CHTR2BTRPV1CYP3A4MEN1
Dimethylamine SCHEMBL7661486 0.81 HTR2C (0.70) DNMT1DNMT3AHTR2CHTR2BDNMT3L
SCHEMBL3807061 0.81 HTR2C (0.73) DNMT1DNMT3AHTR2CHTR2BDNMT3L
SCHEMBL7371691 0.81 HTR2C (0.59) DNMT1DNMT3ACLK1HTR2CHTR2B
SCHEMBL7371124 0.81 FADS1 (0.67) HTR2CHTR2BTRPV1GSK3AGSK3B
SCHEMBL7447310 0.80 HTR2C (0.67) HTR2CHTR2BTRPV1GSK3AGSK3B
SCHEMBL7447576 0.80 HTR2C (0.63) HTR2CHTR2BTRPV1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003737-A1 PHENYL UREA AND PHENYL THIOUREA DERIVATIVES AS HFGAN72 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2000-05-31 EP disclosed
WO-1999009024-A1 PHENYL UREA AND PHENYL THIOUREA DERIVATIVES AS HFGAN72 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1999-02-25 WO disclosed