SCHEMBL740465

SCHEMBL740465

CN1CCC(C#CC(=O)NC2CCCCC2(N)C(=O)c2cc3cc(Cl)ccc3[nH]2)CC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 7/20 0.48
HRH3 Q9Y5N1 5/20 0.48
HRH1 P35367 1/20 0.43
CYP51A1 Q16850 1/20 0.42
F10 P00742 8/20 0.40
F2 P00734 4/20 0.40
PYGL P06737 3/20 0.40
SMYD3 Q9H7B4 1/20 0.40
PYGM P11217 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741493 0.86 SMYD3 (0.45) HRH4HRH3CYP51A1PYGLSMYD3
SCHEMBL742520 0.84 HRH4 (0.44) HRH4HRH3HRH1CYP51A1F10
SCHEMBL741864 0.82 SMYD3 (0.42) CYP51A1PYGLSMYD3PYGM
Hydrochloric Acid SCHEMBL741427 0.82 HRH4 (0.48) HRH4HRH3HRH1CYP51A1F10
SCHEMBL4093939 0.81 F10 (0.57) HRH4HRH3HRH1F10F2
SCHEMBL5902829 0.81 F10 (0.57) HRH4HRH3HRH1F10F2
Hydrochloric Acid SCHEMBL743530 0.78 HRH3 (0.45) HRH4HRH3HRH1CYP51A1F10
Hydrochloric Acid SCHEMBL742844 0.76 F10 (0.50) F10F2
Hydrochloric Acid SCHEMBL739327 0.76 F10 (0.52) F10F2
Hydrochloric Acid SCHEMBL741709 0.76 F10 (0.43) HRH4HRH3HRH1CYP51A1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431370-B1 Monoacylated 1,2-diaminocycloalkanes DAIICHI SANKYO CO LTD (JP) 2013-06-19 EP disclosed
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed
US-7935824-B2 Ethylenediamine derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2011-05-03 US disclosed