SCHEMBL741493

SCHEMBL741493

CC#CC(=O)NC1CCCCC1(N)C(=O)c1cc2cc(Cl)ccc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.45
PYGL P06737 15/20 0.43
CYP51A1 Q16850 1/20 0.42
HRH4 Q9H3N8 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
F7 P08709 1/20 0.40
F3 P13726 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741864 0.88 SMYD3 (0.42) SMYD3PYGLCYP51A1F7F3
SCHEMBL740465 0.86 HRH4 (0.48) SMYD3PYGLCYP51A1HRH4HRH3
SCHEMBL742520 0.84 HRH4 (0.44) PYGLCYP51A1HRH4HRH3
Hydrochloric Acid SCHEMBL741885 0.80 CNR1 (0.47) SMYD3PYGLCYP51A1
Hydrochloric Acid SCHEMBL743335 0.80 SMYD3 (0.46) SMYD3PYGLCYP51A1
SCHEMBL739788 0.79 SMYD3 (0.51) SMYD3PYGLCYP51A1HRH4HRH3
Hydrochloric Acid SCHEMBL743530 0.78 HRH3 (0.45) SMYD3PYGLCYP51A1HRH4HRH3
Hydrochloric Acid SCHEMBL741745 0.78 SMYD3 (0.50) SMYD3PYGLCYP51A1HRH4HRH3
Hydrochloric Acid SCHEMBL742480 0.78 SMYD3 (0.41) SMYD3PYGLCYP51A1
Hydrochloric Acid SCHEMBL742479 0.78 SMYD3 (0.41) SMYD3PYGLCYP51A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431370-B1 Monoacylated 1,2-diaminocycloalkanes DAIICHI SANKYO CO LTD (JP) 2013-06-19 EP disclosed
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed
US-7935824-B2 Ethylenediamine derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2011-05-03 US disclosed