SCHEMBL7405261

SCHEMBL7405261

CC(=O)SC[C@H](C(=O)N[C@@H](Cc1cc2ccccc2o1)C(=O)O)C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.53
PSMB5 P28074 2/20 0.44
PSMB8 P28062 1/20 0.44
FCER2 P06734 2/20 0.44
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 3/20 0.37
ACE P12821 3/20 0.36
MME P08473 3/20 0.35
MMP1 P03956 1/20 0.35
MMP3 P08254 1/20 0.35
TACR1 P25103 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
CPA1 P15085 1/20 0.35
ACE2 Q9BYF1 1/20 0.35
LMNA P02545 2/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7405258 1.00 PIN1 (0.53) PIN1PSMB5PSMB8FCER2NPC1
SCHEMBL7417976 0.85 PIN1 (0.57) PIN1PSMB5PSMB8FCER2NPC1
SCHEMBL7408168 0.85 PIN1 (0.57) PIN1PSMB5PSMB8FCER2NPC1
SCHEMBL7408164 0.85 PIN1 (0.57) PIN1PSMB5PSMB8FCER2NPC1
SCHEMBL7416436 0.81 MME (0.51) FCER2ACEMMEMMP1MMP3
SCHEMBL7419934 0.80 MME (0.53) PIN1PSMB5MEN1KMT2AACE
SCHEMBL7405264 0.78 ACE (0.39) FCER2MEN1KMT2AACEMME
SCHEMBL7407660 0.75 ACE (0.53) ACEMMECPA1ACE2
SCHEMBL7407664 0.75 ACE (0.53) ACEMMECPA1ACE2
SCHEMBL7409095 0.75 ACE (0.53) ACEMMECPA1ACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5414013-A Enzyme inhibitors E. R. SQUIBB & SONS, INC. (US) 1995-05-09 US disclosed
US-5414017-A Cardiovascular agents E. R. SQUIBB & SONS, INC. (US) 1995-05-09 US disclosed
EP-0449523-B1 Mercapto- or acylthio-trifluoromethyl amide derivatives and their use SQUIBB & SONS INC (US) 1994-08-17 EP disclosed
US-5223516-A Endopeptidase inhibitors E. R. SQUIBB & SONS, INC. (US) 1993-06-29 US disclosed
EP-0449523-A1 Mercapto- or acylthio-trifluoromethyl amide derivatives and their use E.R. SQUIBB & SONS, INC. (US) 1991-10-02 EP disclosed