SCHEMBL7405303

SCHEMBL7405303

C=CC(NC(=O)OCc1ccccc1)OC(C=C)NC(=O)OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 2/20 0.55
ATM Q13315 1/20 0.51
TGM2 P21980 1/20 0.51
CTSK P43235 3/20 0.49
TACR1 P25103 2/20 0.49
LMNA P02545 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CTSL P07711 2/20 0.48
CTSS P25774 2/20 0.48
ELANE P08246 1/20 0.48
CTSB P07858 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A2 P05177 1/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22754646 0.84 ATM (0.54) CTRB1ATMCTSKCTSLCTSS
SCHEMBL8173806 0.83 CTRB1 (0.54) CTRB1ATMTGM2CTSKTACR1
SCHEMBL937972 0.83 ATM (0.57) CTRB1ATMCTSKCTSLCTSS
SCHEMBL8101657 0.83 CTRB1 (0.54) CTRB1ATMTGM2CTSKTACR1
SCHEMBL7372388 0.83 CTRB1 (0.54) CTRB1ATMTGM2CTSKTACR1
SCHEMBL937973 0.83 ATM (0.57) CTRB1ATMCTSKCTSLCTSS
SCHEMBL14769904 0.83 CTRB1 (0.54) CTRB1ATMTGM2CTSKTACR1
SCHEMBL22118319 0.83 CTRB1 (0.54) CTRB1ATMTGM2CTSKTACR1
SCHEMBL14396693 0.82 CTSS (0.55) CTRB1ATMCTSKCTSLCTSS
SCHEMBL6712580 0.82 CTRB1 (0.59) CTRB1CTSKTACR1CTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5914313-A ANTIBIOTICS MERCK & CO., INC. (US) 1999-06-22 US disclosed
US-5741775-A ANTIBIOTIC AND ANTIFUNGAL AGENTS MERCK & CO., INC. (US) 1998-04-21 US disclosed
EP-0697879-A4 CYCLOHEXAPEPTIDYL AMINOALKYL ETHERS MERCK & CO INC (US) 1998-01-14 EP disclosed
EP-0697879-A1 CYCLOHEXAPEPTIDYL AMINOALKYL ETHERS MERCK & CO. INC. (US) 1996-02-28 EP disclosed
WO-1994025045-A1 CYCLOHEXAPEPTIDYL AMINOALKYL ETHERS MERCK & CO., INC. (US) 1994-11-10 WO disclosed