SCHEMBL740648

SCHEMBL740648

CC(C(=O)O)C1=C(c2ccc(Cl)c(Cl)c2)c2sc3c(c2CN1C)CCCC3

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 2/20 0.41
AKR1C3 P42330 3/20 0.39
AKR1C2 P52895 3/20 0.39
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
APP P05067 1/20 0.36
SLC6A2 P23975 3/20 0.34
SLC6A3 Q01959 3/20 0.34
TP53 P04637 1/20 0.33
THRB P10828 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PTGS2 P35354 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
EEF2K O00418 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3475686 0.81 KMT2A (0.39) SLC22A12SLC6A2SLC6A3TP53THRB
SCHEMBL740861 0.68 AKR1C3 (0.35) AKR1C3AKR1C2PSEN1PSEN2APH1B
SCHEMBL14926951 0.61 ALDH1A1 (0.40) APPTP53SMN1; SMN2KDM4EKMT2A
SCHEMBL3477086 0.61 ALDH1A1 (0.37) PTGS2KDM4EMEN1KMT2A
SCHEMBL31240209 0.59 AKR1C3 (0.69) AKR1C3AKR1C2PSEN1PSEN2APH1B
SCHEMBL1512537 0.59 AKR1C3 (0.69) AKR1C3AKR1C2PSEN1PSEN2APH1B
SCHEMBL1590709 0.59 AKR1C3 (0.69) AKR1C3AKR1C2PSEN1PSEN2APH1B
SCHEMBL23692158 0.58 AKR1C3 (0.52) AKR1C3AKR1C2PSEN1PSEN2APH1B
SCHEMBL9444855 0.57 AKR1C3 (0.65) AKR1C3AKR1C2PSEN1PSEN2APH1B
SCHEMBL13235896 0.56 AKR1C3 (0.55) AKR1C3AKR1C2PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430029-A1 THIENO [2, 3-B]PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS Katholieke Universiteit Leuven (BE) 2012-03-21 EP disclosed
WO-2010130842-A1 THIENO [2, 3-B] PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2010-11-18 WO disclosed