SCHEMBL7406708

SCHEMBL7406708

N#Cc1ccc(N2CCCNC2=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.49
KDM4E B2RXH2 1/20 0.42
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.41
RPS6KA2 Q15349 1/20 0.39
CYP11B2 P19099 1/20 0.38
ELANE P08246 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
CMA1 P23946 2/20 0.38
CTSG P08311 1/20 0.38
GRM2 Q14416 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
CHRNA10 Q9GZZ6 1/20 0.36
CHRNA9 Q9UGM1 1/20 0.36
ALOX5 P09917 1/20 0.36
F10 P00742 1/20 0.36
PGR P06401 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275896 0.95 HTR1A (0.47) HTR1AKDM4ETP53POLBHRH3
SCHEMBL2713004 0.89 KDM4E (0.49) HTR1AKDM4ETP53POLBCYP11B2
SCHEMBL7282701 0.85 KDM4E (0.45) HTR1AKDM4ETP53POLBHRH3
Bicarbonate SCHEMBL8574872 0.81 CA1 (0.42) HTR1AKDM4ETP53POLBCYP11B2
Bicarbonate SCHEMBL8574878 0.81 CA1 (0.42) HTR1AKDM4ETP53POLBCYP11B2
SCHEMBL14491992 0.80 DDB1 (0.53) HTR1AKDM4ETP53POLBCMA1
Bicarbonate SCHEMBL8574870 0.80 CA1 (0.41) HTR1AKDM4ETP53POLBELANE
SCHEMBL8286230 0.79 SMN1; SMN2 (0.54) KDM4EPOLBELANECMA1CTSG
Hydrochloric Acid SCHEMBL5314439 0.79 DDB1 (0.51) HTR1AKDM4ETP53POLBCMA1
SCHEMBL1259982 0.79 ALDH1A1 (0.46) KDM4ETP53POLBCMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0715623-B1 PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 1998-09-09 EP disclosed
US-5489594-A ANTICOAGULANTS G. D. SEARLE & CO. (US) 1996-02-06 US disclosed
US-5430043-A Platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1995-07-04 US disclosed
WO-1995006038-A1 PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1995-03-02 WO disclosed