SCHEMBL740673

SCHEMBL740673

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](N)CNS(=O)(=O)c3ccc(OC)cc3)C2)nc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
KCNH2 Q12809 5/20 0.45
CYP3A4 P08684 1/20 0.43
ALDH1A1 P00352 6/20 0.43
HRH1 P35367 2/20 0.43
CYP2D6 P10635 1/20 0.43
CHRM1 P11229 1/20 0.42
PKM P14618 1/20 0.42
MAPT P10636 5/20 0.42
POLB P06746 2/20 0.41
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740674 1.00 GAA (0.47) GAAKCNH2CYP3A4ALDH1A1HRH1
SCHEMBL740672 1.00 GAA (0.47) GAAKCNH2CYP3A4ALDH1A1HRH1
SCHEMBL739744 0.94 HRH1 (0.45) GAAKCNH2ALDH1A1HRH1CYP2D6
SCHEMBL739743 0.94 HRH1 (0.45) GAAKCNH2ALDH1A1HRH1CYP2D6
SCHEMBL739745 0.94 HRH1 (0.45) GAAKCNH2ALDH1A1HRH1CYP2D6
SCHEMBL741326 0.93 KCNH2 (0.41) GAAKCNH2CYP3A4ALDH1A1HRH1
SCHEMBL741324 0.93 KCNH2 (0.41) GAAKCNH2CYP3A4ALDH1A1HRH1
SCHEMBL741325 0.93 KCNH2 (0.41) GAAKCNH2CYP3A4ALDH1A1HRH1
SCHEMBL741653 0.93 L3MBTL1 (0.43) GAAKCNH2CYP3A4ALDH1A1HRH1
SCHEMBL741655 0.93 L3MBTL1 (0.43) GAAKCNH2CYP3A4ALDH1A1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed