SCHEMBL740731

SCHEMBL740731

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](N)CNC(=O)c3cccc(OC)c3)C2)nc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.44
KCNH2 Q12809 5/20 0.44
HRH1 P35367 3/20 0.44
CYP2D6 P10635 1/20 0.44
CHRM1 P11229 1/20 0.44
PREP P48147 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CYP3A4 P08684 1/20 0.40
TP53 P04637 1/20 0.39
MCHR1 Q99705 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740733 1.00 ADORA2A (0.44) ADORA2AKCNH2HRH1CYP2D6CHRM1
SCHEMBL740732 1.00 ADORA2A (0.44) ADORA2AKCNH2HRH1CYP2D6CHRM1
SCHEMBL738939 0.94 HRH1 (0.45) ADORA2AKCNH2HRH1CYP2D6CHRM1
SCHEMBL738938 0.94 HRH1 (0.45) ADORA2AKCNH2HRH1CYP2D6CHRM1
SCHEMBL738937 0.94 HRH1 (0.45) ADORA2AKCNH2HRH1CYP2D6CHRM1
SCHEMBL739530 0.92 OPRK1 (0.45) ADORA2AKCNH2HRH1CYP2D6CHRM1
SCHEMBL739531 0.92 OPRK1 (0.45) ADORA2AKCNH2HRH1CYP2D6CHRM1
SCHEMBL739790 0.92 KCNH2 (0.47) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL739791 0.92 KCNH2 (0.47) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL739789 0.92 KCNH2 (0.47) KCNH2HRH1CYP2D6CHRM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed